Monday June 8, 2015 |
| Session Chair: |
Prof. Gilbert KIRSCH (UNIVERSITÉ DE LORRAINE, Metz, France) |
09:00 | Opening |
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09:30 | PL01 - Photoreactive Heterocycles and Natural Product Derivatives |
Prof. Dr Thomas LINDEL (TECHNICAL UNIVERSITY OF BRAUNSCHWEIG, Braunschweig, Germany) |
10:25 | Coffee Break |
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| Session Chair: |
Prof. Mercedes ÁLVAREZ (UNIVERSITY OF BARCELONA, Barcelona, Spain) |
10:55 | PL02 - Targeting DNA Methylation: a Medicinal Chemistry Approach |
Prof. Antonello MAI (UNIVERSITY OF ROME "LA SAPIENZA", Rome, Italy) |
11:50 | IL01 - Synthetic Explorations in Small-ring Azaheterocyclic Chemistry and Development of Novel Bioactive Heterocycles |
Prof. Matthias D'HOOGHE (GHENT UNIVERSITY, Ghent, Belgium) |
12:20 | OC01 - Heterocycle-Peptide Hybrids: Synthesis, Conformational Analysis, and Utilization in Medicinal Chemistry |
Mr Luca GENTILUCCI (UNIVERSITA DI BOLOGNA, Bologna, Italy) |
12:35 | Lunch |
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| Session Chair: |
Prof. Yves FORT (UNIVERSITÉ DE LORRAINE, Nancy, France) |
14:00 | PL03 - The Importance of Heterocycles in Agrochemistry: Fungicides as a Case Study |
Dr Harald WALTER (SYNGENTA CROP PROTECTION AG BASEL, Basel, Switzerland) |
14:55 | IL02 - Synthesis of Biorelevant Heterocycles with N-heterocyclic Carbenes |
Prof. Andreas SCHMIDT (TECHNICAL UNIVERSITY CLAUSTHAL, Clausthal-Zellerfeld, Germany) |
15:25 | OC02 - Exploiting the Zincke Reaction to Produce Sophisticated Heptamethine Dyes |
Dr Robert SMITH (UNIVERSITY OF CENTRAL LANCASHIRE, Prestoin, United Kingdom) |
15:40 | OC03 - Diverse Synthesis of Natural Product Inspired Fused and Spiro-Heterocyclic Scaffolds via Ring Distortion And Construction Strategy |
Prof. Subhabrata SEN (SHIV NADAR UNIVERSITY, Gautam Budh nagar, India) |
15:55 | OC04 - Novel Cross-Conjugated Dienones Based on 4-Piperidone Moiety: Synthesis and Antitumor Properties |
Dr Mikhail MAKAROV (NESMEYANOV INSTITUTE OF ORGANOELEMENT COMPOUNDS OF RAS, Moscow, Russia) |
16:10 | Coffee Break and Poster Session 1 |
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18:00 | Welcome Reception (in the Exhibition area) |
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Tuesday June 9, 2015 |
| Session Chair: |
Dr Stéphanie HESSE (UNIVERSITÉ DE LORRAINE, Metz, France) |
09:00 | PL04 - Non Noble Metal Catalysis for Making Precious Molecules |
Prof. Matthias BELLER (UNIVERSITY OF ROSTOCK, Rostock, Germany) |
09:55 | IL03 - Synthesis of Novel Alpha7-nAchR Ligands: from an Idea to in Rodent Results for Alzheimer [18F] TEP Imaging |
Prof. Sylvain ROUTIER (UNIVERSITÉ D'ORLÉANS, Orléans, France) |
10:25 | OC05 - Recent Advances in the Total Synthesis of Phormidolides B and C |
Mr Alejandro GIL ESCOLANO (IRB BARCELONA, Barcelona, Spain) |
10:40 | Coffee Break |
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| Session Chair: |
Prof. Patrick CHAIMBAULT (UNIVERSITÉ DE LORRAINE, Metz, France) |
11:10 | PL05 - Metal Catalysis for Heteroarene Synthesis |
Prof. Michael GREANEY (THE UNIVERSITY OF MANCHESTER, Manchester, United Kingdom) |
12:05 | IL04 - New Methods in Thioamide Chemistry |
Dr Mike PORTER (UNIVERSITY COLLEGE LONDON, London, United Kingdom) |
12:35 | Lunch |
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| Session Chair: |
Prof. Ferenc FULOP (UNIVERSITY OF SZEGED, Szeged, Hungary) |
14:00 | PL06 - The Discovery and Development of the HIV Intergrase Inhibitors Dolutegravir and Cabotegravir |
Dr Brian JOHNS (GLAXOSMITHKLINE, NC, United States) |
14:55 | IL05 - Are Generic Drugs Only a Copy_and_Paste Products? |
Prof. Stanislav RADL (ZENTIVA, Prague, Czech Republic) |
15:25 | OC06 - An Original Domino Radical Cyclisation/Smiles Rearrangement Combination: Application to the Synthesis of Indolo[2,3-b]Quinoline-Type Derivatives |
Dr. Stéphane GERARD (UNIVERSITÉ DE REIMS - CHAMPAGNE-ARDENNE, REIMS, France) |
15:40 | OC07 - Palladium-Catalyzed Cross-Coupling Reactions in the Asymmetric Synthesis of Pyrrolo[1,2-b]Isoquinolines |
Prof. Nuria SOTOMAYOR (UNIVERSIDAD DEL PAÍS VASCO / EUSKAL HERRIKO UNIBERTSITATEA, Leioa - Bizkaia, Spain) |
15:55 | OC08 - Synthesis of Long Regioregular Dialkyl-Substituted Alpha-Oligofurans |
Dr Edward KORSHIN (THE WEIZMANN INSTITUTE OF SCIENCE, Rehovot, Israel) |
16:10 | Coffee Break and Poster Session 2 |
|
Wednesday June 10, 2015 |
| Session chair: |
Prof. John JOULE (UNIVERSITY OF MANCHESTER, Manchester, United Kingdom) |
09:00 | PL07 - Bronsted Acid and Metal-catalyzed Reactions in the Synthesis of Heterocycles |
Prof. Esther LETE (UNIVERSIDAD DEL PAÍS VASCO, Bilbao, Spain) |
09:55 | IL06 - Utilization of Hypervalent Iodonium Reagents for the Construction and Functionalization of Heterocyclic Molecules |
Dr Zoltan NOVAK (EÖTVÖS UNIVERSITY, Budapest, Hungary) |
10:25 | OC09 - Synthesis of Agrochemistry-Related F-Heterocycles from Novel Fluorinated Diazoalkanes |
Dr Pavel MYKHAILIUK (ENAMINE, Kyiv, Ukraine) |
10:40 | Coffee Break |
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| Session Chair: |
Dr Harald WALTER (SYNGENTA CROP PROTECTION AG BASEL, Basel, Switzerland) |
11:15 | OC10 - Flavylium-Based Pigments – “Click” Synthesis & Biological Relevance |
Dr Stefan CHASSAING (ITAV, Toulouse, France) |
11:30 | OC11 - Synthesis of 7-(2-Aminophenyl)- and 7-(4-Aminophenyl)Guanine, DNA Adducts Derived from the Phenylnitrenium Ion |
Prof. Igor LINHART (UNIVERSITY OF CHEMISTRY AND TECHNOLOGY, Prague, Czech Republic) |
11:45 | OC12 - Heterocyclic Coumarine Analogs as Zinc Metalloprotease Inhibitors |
Mr Peteris TRAPENCIERIS (LATVIAN INSTITUTE OF ORGANIC SYNTHESIS, RIGA, Latvia) |
12:00 | Lunch |
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| Session chair: |
Prof. Milan POTACEK (MASARYK UNIVERSITY, Brno, Czech Republic) |
13:30 | IL07 - Silicon-Containing Tetrahydrocyclopenta[C]Acridine Derivatives as CDKs Inhibitors: Design, Organometallic Synthesis, Metabolic Stability And Optimization |
Prof. Philippe BELMONT (UNIVERSITY PARIS DESCARTES, Paris, France) |
14:00 | OC13 - Synthesis of Imidazo-Pyrrolo-Pyrazines/Diazepines/Diazocines via Domino Ugi/Micheal Reaction and Silver-Catalyzed Heteroannulation |
Mr Zhenghua LI (KU LEUVEN, Leuven, Belgium) |
14:15 | OC14 - Synthesis and Antifungal Activity of N-Acyl Derivatives of 1,4-Benzoxazin- and 1,4-Benzoxazepin-3-ONES |
Mrs Agata GOSZCZYNSKA (WEST POMERANIAN UNIVERSITY OF TECHNOLOGY, SZCZECIN, Szczecin, Poland) |
14:30 | OC15 - Mixed Cu(II) Cu(I) Complexes with Bioheterocycles as the Platform for Construction of Novel Anticancer Agents |
Ms Olga KRASNOVSKAYA (MOSCOW STATE UNIVERSITY, Moscow, Russia) |
14:45 | Coffee Break |
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16:00 | Excursions |
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19:00 | Banquet |
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Thursday June 11, 2015 |
| Session chair: |
Prof. Henk VAN DER PLAS (UNIVERSITY OF WAGENINGEN, Wageningen, The Netherlands) |
09:00 | PL08 - Heterocycles Derived from Natural Products in Management of Multidrug Resistance |
Prof. Ahcene BOUMENDJEL (UNIVERSITÉ JOSEPH FOURIER, La Tronche, France) |
09:55 | IL08 - At the Crossroads of Chemistry and Biology: Inhibiting Protein Kinase CK2 by Heterocyclic Small Molecules |
Prof. Marc LE BORGNE (UNIVERSITÉ CLAUDE BERNARD LYON 1, Lyon, France) |
10:25 | Coffee Break |
|
| Session chair: |
Prof. Jan BERGMAN (KAROLINSKA INSTITUTE, Huddinge, Sweden) |
11:00 | IL09 - Overcoming Resistance with beta-Lactams |
Dr Eric DESARBRE (BASILEA PHARMACEUTICA, Basel, Switzerland) |
11:30 | OC16 - Discovery Of Novel Thieno[3,2-b]Pyrrole 5-Carboxamides as Potent Inhibitors of Chikungunya Virus (CHIKV) |
Mr Kuan Chieh CHING (NATIONAL UNIVERSITY OF SINGAPORE, Singapore, Singapore) |
11:45 | Closing |
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